Structure-activity relationships (SAR) analysis forms the bedrock in drug discovery. By altering the chemical structure of a lead compound and quantifying the resulting biological activity, researchers determine the key structural features responsible for efficacy. This understanding guides further development of novel therapeutic agents with impro

Pharmacological profiling represents a crucial/essential/fundamental step in the development/synthesis/design of novel drug candidates. This process involves/encompasses/includes a comprehensive/thorough/systematic assessment of a drug's pharmacological/therapeutic/biochemical properties, aiming to elucidate/determine/identify its mechanism of acti